J. Med. Chem., 49 (7), 2339 -2352, 2006.
Screening for Cardiovascular Safety: A Structure-Activity Approach for Guiding Lead Selection of Melanin Concentrating Hormone Receptor 1 Antagonists
Philip R. Kym ...
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http://pubs.acs.org/cgi-bin/abstract.cgi/jmcmar/2006/49/i07/abs/jm0512286.html