Discovery and Optimization of Anthranilic Acid Sulfonamides as Inhibitors of Methionine Aminopeptidase-2: A Structural Basis for the Reduction of Albumin Binding
George S. Sheppard,* Jieyi Wang, Megumi Kawai, Steve D. Fidanze, Nwe Y. BaMaung, Scott A. Erickson, David M. Barnes, Jason S. Tedrow, Lawrence Kolaczkowski, Anil Vasudevan, David C. Park, Gary T. Wang, William J. Sanders, Robert A. Mantei, Fabio Palazzo, Lora Tucker-Garcia, Pingping Lou, Qian Zhang, Chang H. Park, Ki H. Kim, Andrew Petros, Edward Olejniczak, David Nettesheim, Phillip Hajduk, Jack Henkin, Richard Lesniewski, Steven K. Davidsen, and Randy L. Bell
J. Med. Chem., 2006, 49 (13), pp 3832–3849
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http://dx.doi.org/10.1021/jm0601001