Bioorganic & Medicinal Chemistry Letters
Volume 15, Issue 8, 15 April 2005, Pages 2129-2134
Potent 1,3,4-trisubstituted pyrrolidine CCR5 receptor antagonists: effects of fused heterocycles on antiviral activity and pharmacokinetic properties
Dooseop Kima, Liping Wang, Jeffrey J. Hale, Christopher L. Lynch, Richard J. Budhu, Malcolm MacCoss, Sander G. Mills, Lorraine Malkowitz, Sandra L. Gould, Julie A. DeMartino, Martin S. Springer, Daria Hazudac, Michael Millerc, Joseph Kesslerc, Renee C. Hrinc, Gwen Carverc, Anthony Carellac, Karen Henryc, Janet Linebergerc, William A. Schleifc and Emilio A. Eminic
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http://dx.doi.org/10.1016/j.bmcl.2005.02.030