+++J. Med. Chem. - часть 2

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1) Antagonists of the Calcium Receptor I. Amino Alcohol-Based Parathyroid Hormone Secretagogues
Robert W. Marquis, Amparo M. Lago, James F. Callahan, Robert E. Lee Trout, Maxine Gowen, Eric G. DelMar, Bradford C. Van Wagenen, Sarah Logan, Scott Shimizu, John Fox, Edward F. Nemeth, Zheng Yang, Theresa Roethke, Brian R. Smith, Keith W. Ward, John Lee, Richard M. Keenan and Pradip Bhatnagar
J. Med. Chem. 2009, 52 (13), pp 3982–3993

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http://dx.doi.org/10.1021/jm900364m

2) Synthesis of Novel 2-Alkoxy-3-amino-3-arylpropan-1-ols and 5-Alkoxy-4-aryl-1,3-oxazinanes with Antimalarial Activity
Matthias D’hooghe, Stijn Dekeukeleire, Karen Mollet, Carmen Lategan, Peter J. Smith, Kelly Chibale and Norbert De Kimpe
J. Med. Chem. 2009, 52 (13), pp 4058–4062

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http://dx.doi.org/10.1021/jm9002632

3) Synthesis and Evaluation of Sphingosine Analogues as Inhibitors of Sphingosine Kinases
Lingkai Wong, Sheryl S. L. Tan, Yulin Lam and Alirio J. Melendez
J. Med. Chem. 2009, 52 (12), pp 3618–3626

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http://dx.doi.org/10.1021/jm900121d

4) Vibriobactin Antibodies: A Vaccine Strategy
Raymond J. Bergeron, Neelam Bharti, Shailendra Singh, James S. McManis, Jan Wiegand and Linda G. Green
J. Med. Chem. 2009, 52 (12), pp 3801–3813

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http://dx.doi.org/10.1021/jm900119q

5) Discovery of Highly Potent and Selective Biphenylacylsulfonamide-Based β3-Adrenergic Receptor Agonists and Evaluation of Physical Properties as Potential Overactive Bladder Therapies: Part 5
Kouji Hattori, Susumu Toda, Masashi Imanishi, Shinji Itou, Yutaka Nakajima, Kenichi Washizuka, Takanobu Araki, Hitoshi Hamashima, Yasuyo Tomishima, Minoru Sakurai, Shigeo Matsui, Emiko Imamura, Koji Ueshima, Takao Yamamoto, Nobuhiro Yamamoto, Hirofumi Ishikawa, Keiko Nakano, Naoko Unami, Kaori Hamada, Yasuhiro Matsumura and Fujiko Takamura
J. Med. Chem. 2009, 52 (9), pp 3063–3072

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http://dx.doi.org/10.1021/jm9000709

6) Synthesis and Structure−Activity Relationships of Long-acting β2 Adrenergic Receptor Agonists Incorporating Arylsulfonamide Groups
Panayiotis A. Procopiou, Victoria J. Barrett, Nicola J. Bevan, Keith Biggadike, Peter R. Butchers, Diane M. Coe, Richard Conroy, Dean D. Edney, Rita N. Field, Alison J. Ford, Stephen B. Guntrip, Brian E. Looker, Iain M. McLay, Michael J. Monteith, Valerie S. Morrison, Peter J. Mutch, Stephen A. Richards, Rosemary Sasse and Claire E. Smith
J. Med. Chem. 2009, 52 (8), pp 2280–2288

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http://dx.doi.org/10.1021/jm801016j

7) N6-Cycloalkyl- and N6-Bicycloalkyl-C5′(C2′)-modified Adenosine Derivatives as High-Affinity and Selective Agonists at the Human A1 Adenosine Receptor with Antinociceptive Effects in Mice
Palmarisa Franchetti, Loredana Cappellacci, Patrizia Vita, Riccardo Petrelli, Antonio Lavecchia, Sonja Kachler, Karl-Norbert Klotz, Ida Marabese, Livio Luongo, Sabatino Maione and Mario Grifantini
J. Med. Chem. 2009, 52 (8), pp 2393–2406

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http://dx.doi.org/10.1021/jm801456g

8 ) N-(4-(4-(2,3-Dichloro- or 2-methoxyphenyl)piperazin-1-yl)butyl)heterobiarylcarboxamides with Functionalized Linking Chains as High Affinity and Enantioselective D3 Receptor Antagonists
Amy Hauck Newman, Peter Grundt, George Cyriac, Jeffrey R. Deschamps, Michelle Taylor, Rakesh Kumar, David Ho and Robert R. Luedtke
J. Med. Chem. 2009, 52 (8), pp 2559–2570

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http://dx.doi.org/10.1021/jm900095y

9) Synthesis and Pharmacological Characterization of β2-Adrenergic Agonist Enantiomers: Zilpaterol
Christopher Kern, Thorsten Meyer, Serge Droux, Dieter Schollmeyer and Christian Miculka
J. Med. Chem. 2009, 52 (6), pp 1773–1777

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http://dx.doi.org/10.1021/jm801211c

10) Synthesis and in Vitro and in Vivo Evaluation of 18F-Labeled Positron Emission Tomography (PET) Ligands for Imaging the Vesicular Acetylcholine Transporter
Zhude Tu, Simon M. N. Efange, Jinbin Xu, Shihong Li, Lynne A. Jones, Stanley M. Parsons and Robert H. Mach
J. Med. Chem. 2009, 52 (5), pp 1358–1369

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http://dx.doi.org/10.1021/jm8012344

11) Enantioselectivity in Cardioprotection induced by (S)- (−)-2,2-Dimethyl-N-(4′-acetamido-benzyl)-4-spiromorpholone-chromane
Simona Rapposelli, Vincenzo Calderone, Roberto Cirilli, Maria Digiacomo, Cristina Faggi, Francesco La Torre, Mariaelisa Manganaro, Alma Martelli and Lara Testai
J. Med. Chem. 2009, 52 (5), pp 1477–1480

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http://dx.doi.org/10.1021/jm801459f

12) Synthesis, Radiosynthesis, and Biological Evaluation of Carbon-11 and Fluorine-18 Labeled Reboxetine Analogues: Potential Positron Emission Tomography Radioligands for in Vivo Imaging of the Norepinephrine Transporter
Fanxing Zeng, Jiyoung Mun, Nachwa Jarkas, Jeffrey S. Stehouwer, Ronald J. Voll, Gilles D. Tamagnan, Leonard Howell, John R. Votaw, Clinton D. Kilts, Charles B. Nemeroff and Mark M. Goodman
J. Med. Chem. 2009, 52 (1), pp 62–73

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http://dx.doi.org/10.1021/jm800817h

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jm900364m.pdf

jm9000709.pdf

jm900119q.pdf

jm900121d.pdf

jm801016j.pdf

jm801456g.pdf

jm9002632.pdf

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