1) Piperazinyl Glutamate Pyridines as Potent Orally Bioavailable P2Y12 Antagonists for Inhibition of Platelet Aggregation
John J. Parlow*†, Mary W. Burney‡, Brenda L. Case†, Thomas J. Girard‡, Kerri A. Hall‡, Peter K. Harris‡, Ronald R. Hiebsch‡, Rita M. Huff‡, Rhonda M. Lachance‡, Deborah A. Mischke†, Stephen R. Rapp‡, Rhonda S. Woerndle† and Michael D. Ennis
J. Med. Chem., 2010, 53 (5), pp 2010–2037
DOI:
- DOI:
http://dx.doi.org/10.1021/jm901518t
Younis Baqi†, Kerstin Atzler†, Meryem Kse†, Markus Glnzel§‡ and Christa E. Mller
J. Med. Chem., 2009, 52 (12), pp 3784–3793
DOI:
- DOI:
http://dx.doi.org/10.1021/jm9003297