Concise synthesis of ω-fluoroalkylated ketoesters. A building block for the synthesis of six-, seven-, and eight-membered fluoroalkyl substituted 1,2-diaza-3-one heterocycles
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Tetrahedron, 2009 , vol. 65, # 21 p. 4212 - 4219
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http://dx.doi.org/10.1016/j.tet.2009.03.029Rémy C. Lemoinea, , , Ann C. Petersena, †, Lina Settia, Andreas Jekleb, Gabrielle Heilekb, André deRosierb, Changhua Jib, Pamela Berryc, ‡, David M. Rotstein
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http://dx.doi.org/10.1016/j.bmcl.2010.06.135 Emmanuel Pinard*, Alexander Alanine, Daniela Alberati, Markus Bender, Edilio Borroni, Patrick Bourdeaux
J. Med. Chem., 2010, 53 (12), pp 4603–4614
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http://dx.doi.org/10.1021/jm100210p