Development of a Scalable Synthesis of Dipeptidyl Peptidase-4 Inhibitor ABT-279
Todd S. McDermott, Lakshmi Bhagavatula, Thomas B. Borchardt, Kenneth M. Engstrom, Jorge Gandarilla,
Brian J. Kotecki, Albert W. Kruger, Michael J. Rozema, Ahmad Y. Sheikh, Seble H. Wagaw and Steven J. Wittenberger
Org. Process Res. Dev., 2009, 13 (6), pp 1145–1155
- DOI:
http://dx.doi.org/10.1021/op900197r