Akihiko Tanitame, Yoshihiro Oyamada, Keiko Ofuji, Mika Fujimoto, Noritaka Iwai, Yoichi Hiyama, Kenji Suzuki, Synthesis and Antibacterial Activity of a Novel Series of Potent DNA Gyrase Inhibitors. Pyrazole Derivatives, J. Med. Chem., 2004, 47 (14), pp 3693–3696
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http://dx.doi.org/10.1021/jm030394f