Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a
Philip J. Skinner, Martin C. Cherrier, Peter J. Webb, Young-Jun Shin, Tawfik Gharbaoui, Andrew Lindstrom, Vu Hong, Susan Y. Tamura, Huong T. Dang, Cameron C. Pride, Ruoping Chen, Jeremy G. Richman, Daniel T. Connolly, Graeme Semple
Bioorganic & Medicinal Chemistry Letters, Volume 17, Issue 20, 15 October 2007, Pages 5620-5623
- DOI:
http://dx.doi.org/10.1016/j.bmcl.2007.07.101
Michael P. DeNinnoa, Melissa Andrewsa, Andrew S. Bellb, Yue Chena, Cynthia Eller-Zarboa, Nan Eshelbyb, John B. Etiennea,
Dianna E. Moorea, Michael J. Palmerb, Michael S. Vissera, Li J. Yua, William J. Zavadoskia, E. Michael Gibbsa
Bioorganic & Medicinal Chemistry Letters, Volume 19, Issue 9, 1 May 2009, Pages 2537–2541
- DOI:
http://dx.doi.org/10.1016/j.bmcl.2009.03.024